Actelion Pharmaceuticals Ltd v. Mylan Pharmaceuticals Inc.

CourtCourt of Appeals for the Federal Circuit
DecidedMay 13, 2026
Docket24-1641
StatusPublished

This text of Actelion Pharmaceuticals Ltd v. Mylan Pharmaceuticals Inc. (Actelion Pharmaceuticals Ltd v. Mylan Pharmaceuticals Inc.) is published on Counsel Stack Legal Research, covering Court of Appeals for the Federal Circuit primary law. Counsel Stack provides free access to over 12 million legal documents including statutes, case law, regulations, and constitutions.

Bluebook
Actelion Pharmaceuticals Ltd v. Mylan Pharmaceuticals Inc., (Fed. Cir. 2026).

Opinion

Case: 24-1641 Document: 54 Page: 1 Filed: 05/13/2026

United States Court of Appeals for the Federal Circuit ______________________

ACTELION PHARMACEUTICALS LTD, Plaintiff-Appellant

v.

MYLAN PHARMACEUTICALS INC., Defendant-Appellee ______________________

2024-1641 ______________________

Appeal from the United States District Court for the Northern District of West Virginia in No. 1:20-cv-00110- JPB, Judge John Preston Bailey. ______________________

Decided: May 13, 2026 ______________________

LISA GLASSER, Irell & Manella LLP, Newport Beach, CA, argued for plaintiff-appellant. Also represented by JASON SHEASBY, Los Angeles, CA; PHILIP J. WARRICK, Washington, DC.

ERIC THOMAS WERLINGER, Katten Muchin Rosenman LLP, Washington, DC, argued for defendant-appellee. Also represented by TIMOTHY H. GRAY; JITENDRA MALIK, Char- lotte, NC; DEEPRO MUKERJEE, LANCE SODERSTROM, New York, NY; JILLIAN SCHURR-HENDRIX, Dallas, TX. ______________________ Case: 24-1641 Document: 54 Page: 2 Filed: 05/13/2026

Before REYNA, TARANTO, and STOLL, Circuit Judges. TARANTO, Circuit Judge. Actelion Pharmaceuticals Ltd owns U.S. Patent Nos. 8,318,802 and 8,598,227, which describe certain phar- maceutical compositions involving epoprostenol. Epo- prostenol is the active ingredient in Actelion’s hypertension drug Veletri®. Mylan Pharmaceuticals Inc. submitted an abbreviated new drug application (ANDA) to the Food and Drug Administration (FDA) seeking approval to market a generic epoprostenol drug before the expiration of Actelion’s patents. Actelion sued Mylan for patent in- fringement in the Northern District of West Virginia under 35 U.S.C. § 271(e)(2) and 21 U.S.C. § 355(j), alleging that Mylan’s proposed generic drug was covered (literally or un- der the doctrine of equivalents) by certain claims of the ’802 and ’227 patents. The district court found no literal in- fringement, concluding, as most relevant here, that the claim term “a pH of 13 or higher” refers to a pH measured at a temperature standard in the field. The district court further ruled that Actelion was barred from asserting, and had not proved, infringement by an equivalent. Actelion appeals. We now affirm. I A The ’802 and ’227 patents are both titled “Epoprostenol Formulation and Method of Making Thereof.” The ’227 pa- tent issued from a divisional of the application that issued as the ’802 patent, and they share a specification, so we cite only the ’802 patent’s specification. Epoprostenol is a vasodilator and antiplatelet agent that can be used to treat cardiovascular disease. It is un- stable in water and will react with water molecules to form a different compound that lacks epoprostenol’s desirable pharmacological properties. ’802 patent, col. 2, lines 41– 51; col. 2, line 65, through col. 3, line 51. Case: 24-1641 Document: 54 Page: 3 Filed: 05/13/2026

ACTELION PHARMACEUTICALS LTD v. 3 MYLAN PHARMACEUTICALS INC.

The presence of an acid in an aqueous (water-based) solution of epoprostenol rapidly catalyzes this unwanted reaction. Acidic molecules in water can dissociate, intro- ducing hydrogen ions (H+) into the solution, which are also present as a result of water molecules’ own dissociation. Such hydrogen ions often interact with water molecules to form what is represented as a water molecule with an extra hydrogen ion, called hydronium (H3O+). These hydrogen ions or hydronium ions facilitate the degradation of epo- prostenol in water. As catalysts, they are not consumed by the reaction of epoprostenol with water, so even trace amounts can cause continuing breakdown of epoprostenol. See ’802 patent, col. 2, line 65, through col. 3, line 51; J.A. 35–36. The degree of acidity of a solution is commonly ex- pressed using the pH scale. pH is a positive number—the negative of the base-ten logarithm of the concentration of hydrogen ions, that logarithm being a negative number. (For simplicity, we now omit separate mention of hydro- nium ions.) The higher the concentration of hydrogen ions, the lower the pH. Under standard ambient conditions, in- cluding a temperature of 25°C, the pH of pure water is 7, sometimes called neutral pH, with values higher than 7 considered basic and values lower than 7 considered acidic. See ’802 patent, col. 4, lines 62–64; J.A. 31–32. The concentration of hydrogen ions in a given solution can be modified in at least two ways. First, one can add acidic or basic compounds to the solution. An acid, as al- ready noted, will introduce more hydrogen ions into a solu- tion (increasing the concentration, thus lowering the pH), and a base will have the opposite effect, reacting with hy- drogen ions and neutralizing them (decreasing the hydro- gen-ion concentration, thus raising the pH). See ’802 patent, col. 2, lines 56–57; col. 4, line 62, through col. 5, line 21. Second, one can change the temperature of the solu- tion. Increasing the temperature will cause molecules that are susceptible to liberating hydrogen ions (like water) to Case: 24-1641 Document: 54 Page: 4 Filed: 05/13/2026

dissociate more frequently, while decreasing the tempera- ture will do the opposite. See J.A. 35–36. Before the priority date of the ’802 patent and Actelion’s subsequent introduction of Veletri, the FDA ap- proved the marketing of Flolan®, another epoprostenol for- mulation for intravenous administration. ’802 patent, col. 2, lines 41–57. Flolan had three features that mitigated the acid-catalyzed degradation of epoprostenol in water. First, it was stored as a lyophilized (freeze-dried) powder and reconstituted into an aqueous solution (by mixing with liquid diluent) just before it was to be administered. Sec- ond, Flolan included a special diluent for reconstituting the freeze-dried powder that was more basic than typical intra- venous fluids. Third, the reconstituted solution was refrig- erated. See ’802 patent, col. 3, lines 52–67. The ’802 patent states that Flolan’s needs for a special diluent and refrigeration were inconvenient, suggesting the desirability of providing epoprostenol compositions that would be suitably stable even when reconstituted with common commercially available intravenous fluids (which are more acidic than the Flolan diluent) and kept at room temperature (at which hydrogen-ion concentration would be greater than during refrigeration). See ’802 patent, col. 4, lines 1–19. To that end, the inventor designed processes for making lyophilized epoprostenol compositions that “when reconstituted ha[ve] a pH>11,” a pH higher than that of reconstituted Flolan, which is around 10.5. See ’802 patent, col. 4, lines 20–23; col. 3, lines 52–56; col. 7, line 51, through col. 8, line 57. To achieve such a high pH in the reconstituted solution without using Flolan’s basic diluent, the patent discloses creating a highly basic “bulk solution” that includes epoprostenol. The patent discloses adding ar- ginine (a mildly basic amino acid) and sodium hydroxide or other bases to the bulk solution to increase its pH. ’802 patent, col. 4, line 62, through col. 5, line 43. The bulk so- lution is then freeze-dried to yield a powder containing suf- ficient amounts of basic molecules to provide an Case: 24-1641 Document: 54 Page: 5 Filed: 05/13/2026

ACTELION PHARMACEUTICALS LTD v. 5 MYLAN PHARMACEUTICALS INC.

appropriately basic solution when reconstituted with a cer- tain quantity of typical intravenous fluid (e.g., saline). See ’802 patent, col. 5, line 22, through col. 7, line 30.

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